Bioactivity:

GB-110 selectively induces PAR2-mediated intracellular Ca2+ release in HT29 cells with an EC50 of 0.28 _M.�GB-110 is a potent, orally active, and nonpeptidic protease activated receptor 2 (PAR2) agonist.

CAS nr:

1252806-70-4

Purity:

98%

Molecular Weight:

608,77

SMILES:

O=C(C1=CC=NO1)N[C@@H](CC2CCCCC2)C(N[C@@H]([C@@H](C)CC)C(NCC3=CC=CC(C(N4CCC(CN)CC4)=O)=C3)=O)=O

Formula:

C33H48N6O5

Pathway:

Others

Target:

Others