Bioactivity:

PEAQX(NVP-AAM 077) is an effective and orally available NMDA antagonist. It can inhibit human NMDA receptors for 1A/2A(IC50: 270 nM), rather than 1A/2B(29, 600 nM).

CAS nr:

459836-30-7

Purity:

98%

Molecular Weight:

454,2

SMILES:

O=c1c(=O)[nH]c2c(c(C(P(=O)(O)O)N[C@H](c3ccc(Br)cc3)C)ccc2)[nH]1

Formula:

C17H17BrN3O5P

Pathway:

Neuroscience,Neuroscience,Membrane transporter/Ion channel

Target:

NMDAR,iGluR,iGluR