Bioactivity:

EN4 MYC inhibitor is a covalent ligand that targets cysteine 171 (C171) of MYC. It is selective for c-MYC over N-MYC and L-MYC, and inhibits MYC transcriptional activity, downregulates MYC targets, and impairs tumorigenesis.

CAS nr:

1197824-15-9

Purity:

98%

Molecular Weight:

416,47

SMILES:

CCOC1=CC=C(C=C1)OC2=CC=CC=C2NC(=O)C3=CC=C(C=C3)CNC(=O)C=C

Formula:

C25H24N2O4

Pathway:

Cell Cycle/Checkpoint

Target:

c-Myc