A-366 T3624
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
Potent and selective G9a/GLP histone lysine methyltransferase inhibitor (IC50�= 3.3 nM). Exhibits >1000-fold selectivity for G9a/GLP over 21 other methyltransferases. Decreases levels of lysine 9 dimethylation on histone H3 (H3K9Me2) in PC3 cells.
CAS nr:
1527503-11-2
Purity:
98%
Molecular Weight:
329,44
SMILES:
COc1cc2c(cc1OCCCN1CCCC1)N=C(N)C21CCC1
Formula:
C19H27N3O2
Pathway:
Chromatin/Epigenetic,Chromatin/Epigenetic
Target:
Epigenetic Reader Domain,Histone Methyltransferase
