Bioactivity:

Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).

CAS nr:

137565-28-7

Purity:

98%

Molecular Weight:

804

SMILES:

CCCC[C@H](NC(=O)[C@H](CC(C)C)N(C)C(=O)CNC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](N)CC(O)=O)C(C)C)C(N)=O

Formula:

C39H65N9O9

Pathway:

GPCR/G Protein,Neuroscience

Target:

Neurokinin receptor,Neurokinin receptor