Bioactivity:

Amelubant (BIIL 284) is a prodrug of active metabolites BIIL 260 and BIIL 315. Anti-inflammatory activity[1]. Amelubant (BIIL 284) is a potent, oral and long acting LTB4 receptor antagonist, negligibly binds to LTB4 receptor, with Kis of 221 nM and 230 nM

CAS nr:

346735-24-8

Purity:

98%

Molecular Weight:

538,63

SMILES:

CC(C1=CC=C(OCC2=CC(COC3=CC=C(C(NC(OCC)=O)=N)C=C3)=CC=C2)C=C1)(C4=CC=C(O)C=C4)C

Formula:

C33H34N2O5

Pathway:

Immunology/Inflammation

Target:

LTR