ADWX 1 TP2080
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
Potent and selective KV1.3 channel blocker (IC50 values are 0.0019 and 0.65 nM for KV1.3 and KV1.1, respectively). Inhibits CD4+ CCR7- T cell activation. Ameliorates rat experimental autoimmune encephalomyelitis, in a model for multiple sclerosis.
CAS nr:
TP2080
Purity:
98%
Molecular Weight:
4071,86
SMILES:
Formula:
C169H281N57O46S7
Pathway:
Target:
