Bioactivity:

Lintitript is an orally active, competitive, and non-peptide cholecystokinin (CCK1) receptor antagonist (EC50: 6 nM; Ki: 0.2 nM). Lintitript shows > 33-fold selectivity more selective for CCK1 than CCK2 receptors (EC50: 200 nM).

CAS nr:

136381-85-6

Purity:

98%

Molecular Weight:

411,86

SMILES:

O=C(O)CN1C(C(NC2=NC(C3=CC=CC=C3Cl)=CS2)=O)=CC4=C1C=CC=C4

Formula:

C20H14ClN3O3S

Pathway:

GPCR/G Protein

Target:

cholecystokinin