Bioactivity:

SNT-207858 is a selective, blood brain barrier penetrating, potent and orally active antagonist of melanocortin-4 (MC-4) receptor. SNT207858 has an IC50 of 22 nM (binding) and 11 nM (function) on the MC-4 receptor.

CAS nr:

1104080-42-3

Purity:

98%

Molecular Weight:

689,54

SMILES:

[H]Cl.O=C(N1CCCC1)N[C@H](CC2=CC=C(Cl)C=C2Cl)C(N3CCC(C4=NC=CC=C4OC[C@H](N5CCCC5)CC)CC3)=O.[H]Cl

Formula:

C32H45Cl4N5O3

Pathway:

Others

Target:

Others