Bioactivity:

NTRC-824 is >150-fold selectivity for NTS2 over NTS1 (Ki >30 _M). NTRC-824 is an effective, selective, and neurotensin-like nonpeptide neurotensin receptor type 2 (NTS2) antagonist (IC50: 38 nM and a Ki : 202 nM).

CAS nr:

1623002-61-8

Purity:

98%

Molecular Weight:

553,55

SMILES:

CC(C)C[C@@H](C(O)=O)NC(CN1C=C(C(C(F)(F)F)=O)C2=C1C=CC(NS(=O)(C3=CC=C(C)C=C3)=O)=C2)=O

Formula:

C25H26F3N3O6S

Pathway:

Others

Target:

Others