Bioactivity:

MRS2179 is a competitive P2Y1 receptor antagonist (Kb = 100 nM) with no appreciable activity at P2Y2, P2Y4, or P2Y6 at concentrations up to 30 ﾵM, or at P2Y12 and P2Y13. It inhibits ADP-induced platelet shape change and aggregation (pA2 = 6.55) in vitro a

CAS nr:

101204-49-3

Purity:

98%

Molecular Weight:

423,22

SMILES:

O=P(OC1C(COP([O-])(O)=O)OC(N2C=NC3=C(NC)N=CN=C23)C1)([O-])O

Formula:

C11H15N5O9P22-

Pathway:

Target: