Bioactivity:

YM022 is a highly effective and selective gastrin/cholecystokinin (CCK)-B receptor antagonist. YM022 can inhibit gastrin-induced gastric acid secretion and histidine decarboxylase activation in vivo. YM022 shows the Ki values of 68 pM and 63 nM for CCK-B

CAS nr:

145084-28-2

Purity:

98%

Molecular Weight:

516,59

SMILES:

O=C(NC1=CC=CC(C)=C1)N[C@H]2C(N(CC(C3=CC=CC=C3C)=O)C4=CC=CC=C4C(C5=CC=CC=C5)=N2)=O

Formula:

C32H28N4O3

Pathway:

Microbiology/Virology,Immunology/Inflammation

Target:

CCR,CCR