Bioactivity:

ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM. ELN-441958 is highly selective for B1 over B2 receptors.

CAS nr:

913064-47-8

Purity:

98%

Molecular Weight:

501,02

SMILES:

Clc1cccc2c1C(=O)N(C2)c1cccc(c1)C(=O)N1CCC2(CC1)CCN(CC2)c1ccncc1

Formula:

C29H29ClN4O2

Pathway:

GPCR/G Protein

Target:

Bradykinin Receptor