Bioactivity:

TPA-023B is an orally active and high-affinity agonist of the GABAA receptor _2/_3 subtype (Kis: 0.73 nM/2 nM) partial and an antagonist _1 subtype (Ki: 1.8 nM), has non-sedating anxiolytic-like properties.

CAS nr:

425377-76-0

Purity:

98%

Molecular Weight:

391,37

SMILES:

N#CC1=CC=CC(F)=C1C2=CC(C3=CN=C4N3N=CC(C(C)(O)C)=N4)=CC=C2F

Formula:

C21H15F2N5O

Pathway:

Others

Target:

Others