Bioactivity:

BAY-1797 is an orally active and selective P2X4 antagonist (IC50: 211 nM against human P2X4) with anti-nociceptive and anti-inflammatory effects. BAY-1797 displays no or very weak activity on the other P2X ion channels.

CAS nr:

2055602-83-8

Purity:

98%

Molecular Weight:

416,88

SMILES:

C1=CC=C(C=C1)CC(=O)NC2=CC(=C(C=C2)OC3=CC(=CC=C3)Cl)S(=O)(=O)N

Formula:

C20H17ClN2O4S

Pathway:

Membrane transporter/Ion channel,Neuroscience

Target:

P2X Receptor,P2 Receptor