Bioactivity:

Fananserin is an orally bioavailable and selective antagonist of the 5-HT2 receptor (Ki: 0.37 nM for the rat 5-HT2A receptor). It also is an antagonist of dopamine D4 receptor (Ki: 2.93 nM for the human dopamine D4 receptor).

CAS nr:

127625-29-0

Purity:

98%

Molecular Weight:

425,52

SMILES:

FC1=CC=C(N2CCN(CCCN(C3=CC=CC4=C3C5=CC=C4)S5(=O)=O)CC2)C=C1

Formula:

C23H24FN3O2S

Pathway:

Neuroscience,GPCR/G Protein,GPCR/G Protein,Neuroscience

Target:

5-HT Receptor,5-HT Receptor,Dopamine Receptor,Dopamine Receptor