Bioactivity:

CARM1-IN-1 shows high and selective CARM1 inhibition, with lower or no activity against a panel of different PRMTs or HKMTs. In human LNCaP cells, CARM1-IN-1 dose-dependently reduces of the PSA promoter activity.

CAS nr:

T10682

Purity:

98%

Molecular Weight:

591,72

SMILES:

[H]Cl.O=C1/C(CN(CC2=CC=CC=C2)C/C1=C\C3=CC=C(O)C(Br)=C3)=C/C4=CC=C(O)C(Br)=C4

Formula:

C26H22Br2ClNO3

Pathway:

Others

Target:

Others