Bioactivity:

FTI-2153 is a potent and highly selective farnesyltransferase (FTase) inhibitor (IC50: 1.4 nM). FTI-2153 is >3000-fold more potent at blocking H-Ras (IC50, 10 nM) than Rap1A processing.

CAS nr:

344900-92-1

Purity:

98%

Molecular Weight:

466,6

SMILES:

CSCC[C@@H](C(OC)=O)NC(C1=CC=C(CNCC2=CN=CN2)C=C1C3=CC=CC=C3C)=O

Formula:

C25H30N4O3S

Pathway:

Others

Target:

Others