Bioactivity:

NI-57 is an inhibitor of proteins of bromodomain and plant homeodomain finger-containing (BRPF) family, with IC50s of 3.1, 46 and 140 nM for BRPF1, BRPF2 (BRD1) and BRPF3, respectively.

CAS nr:

1883548-89-7

Purity:

98%

Molecular Weight:

383,4

SMILES:

COC1=CC(=CC=C1S(=O)(=O)NC1=CC=C2N(C)C(=O)C(C)=CC2=C1)C#N

Formula:

C19H17N3O4S

Pathway:

Chromatin/Epigenetic

Target:

Epigenetic Reader Domain