Bioactivity:

CPI-360 is a potent, selective, and SAM-competitive EZH1 inhibitor with IC50 of 102.3 nM, >100-fold selectivity over other methyltransferases.

CAS nr:

1802175-06-9

Purity:

98%

Molecular Weight:

437,53

SMILES:

COC1=C(CNC(=O)C2=C(C)N([C@H](C)C3CCOCC3)C3=C2C=CC=C3)C(=O)NC(C)=C1

Formula:

C25H31N3O4

Pathway:

Chromatin/Epigenetic,Apoptosis

Target:

Histone Methyltransferase,Apoptosis