Bioactivity:

MS049 is a potent and selective inhibitor of PRMT4 (IC50 = 34 nM) and PRMT6 (IC50 = 43 nM). It is less active against additional type I PRMTs (IC50s = >130, >220, and 1.6 _M for PRMT1, PRMT3, and PRMT8, respectively) and displays no inhibition against typ

CAS nr:

T4393

Purity:

98%

Molecular Weight:

321,28

SMILES:

Cl.Cl.CNCCN1CCC(CC1)OCc2ccccc2

Formula:

C15H26Cl2N2O

Pathway:

Chromatin/Epigenetic

Target:

Histone Methyltransferase