Bioactivity:

BMS-193885 is a potent, selective, competitive, and brain penetrant neuropeptide Y1 receptor antagonist. With a Ki of 3.3 nM, and has an IC50 of 5.9 nM for hY1. It displays > 100, > 160, > 160 and > 160-fold selectivity over _1, hY2, hY4 and hY5 receptors

CAS nr:

186185-03-5

Purity:

98%

Molecular Weight:

590,71

SMILES:

O=C(C1=C(C)NC(C)=C(C(OC)=O)C1C2=CC=CC(NC(NCCCN3CCC(C4=CC=CC(OC)=C4)CC3)=O)=C2)OC

Formula:

C33H42N4O6

Pathway:

Others

Target:

Others