Bioactivity:

SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors, respectively).

CAS nr:

464930-42-5

Purity:

98%

Molecular Weight:

793,41

SMILES:

Cl.COc1ccc2cc(ccc2c1)S(=O)(=O)N[C@H](CC(=O)N[C@H](Cc1ccc(CN2[C@@H](C)CCC[C@H]2C)cc1)C(=O)N(C)C(C)C)c1ccc2OCOc2c1

Formula:

C42H53ClN4O7S

Pathway:

GPCR/G Protein

Target:

Bradykinin Receptor