Bioactivity:

MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1, and A3 receptors respectively. MRS-1706 is an effective and selective adenosine A2B receptor inverse agonist.

CAS nr:

264622-53-9

Purity:

98%

Molecular Weight:

503,55

SMILES:

O=C(NC1=CC=C(C(C)=O)C=C1)COC2=CC=C(C3=NC(N(CCC)C(N(CCC)C4=O)=O)=C4N3)C=C2

Formula:

C27H29N5O5

Pathway:

Neuroscience,GPCR/G Protein

Target:

Adenosine Receptor,Adenosine Receptor