Bioactivity:

Mardepodect is an effective and selective PDE10A inhibitor (IC50: 0.37 nM). Mardepodect has >1000-fold selectivity over other PDEs. Mardepodect can cross the blood-brain barrier.

CAS nr:

898562-94-2

Purity:

98%

Molecular Weight:

392,45

SMILES:

CN(N=C1C2=CC=C(OCC3=NC4=CC=CC=C4C=C3)C=C2)C=C1C5=CC=NC=C5

Formula:

C25H20N4O

Pathway:

Metabolism

Target:

PDE