Bioactivity:

FSLLRY-NH2 TFA is a is a protease-activated receptor 2 (PAR2) inhibitor.�Reverses taxol-induced mechanical allodynia, heat hyperalgesia and PKC activation in ICR mice.�Blocks ERK activation and collagen production in isolated cardiac fibroblasts.�Also red

CAS nr:

TP1904L

Purity:

98%

Molecular Weight:

910,99

SMILES:

CC(C)C[C@@H](C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC1=CC=C(C=C1)O)C(=O)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@H](CC2=CC=CC=C2)N.O=C(O)C(F)(F)F

Formula:

C41H61F3N10O10

Pathway:

GPCR/G Protein

Target:

Protease-activated Receptor