Tertiapin LQ TP2113
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
Blocker of Kir1.1 channels; displays >250-fold selectivity for Kir1.1 (Kd values are 1.1, 274 and 361 nM for Kir1.1, Kir3.1/3.2 and Kir3.1/3.4 respectively). Derivative of tertiapin-Q.
CAS nr:
TP2113
Purity:
98%
Molecular Weight:
2428,03
SMILES:
Formula:
C106H179N33O24S4
Pathway:
Target:
