Bioactivity:

KZR-504 is a selective inhibitor of immunoproteasome low molecular mass polypeptide 2 (LMP2) (IC50s: 51 nM, 4.274 _M for LMP2 and LMP7, respectively).

CAS nr:

1629052-78-3

Purity:

98%

Molecular Weight:

413,42

SMILES:

O=C(N[C@@H](CO)C(N[C@@H](CC1=CC=CC=C1)C([C@]2(CO2)C)=O)=O)C(N3)=CC=CC3=O

Formula:

C21H23N3O6

Pathway:

Proteases/Proteasome,Ubiquitination

Target:

Proteasome,Proteasome