Bioactivity:

YM-430 is a _1 adrenergic receptor antagonist and a calcium channel antagonist. YM430 could be both an antianginal and antihypertensive agent. YM430 (10(-8)-10(-6) M) inhibited 3,4-diaminopyridine-induced rhythmic contractions with an IC50 value of 59.2 n

CAS nr:

153192-22-4

Purity:

98%

Molecular Weight:

553,61

SMILES:

O=C(C1=C(C)NC(C)=C(C(OCCCCNC[C@H](O)COC2=CC=CC=C2)=O)[C@H]1C3=CC=CC([N+]([O-])=O)=C3)OC

Formula:

C29H35N3O8

Pathway:

Target: