Bioactivity:

GSK1016790A (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial cells.

CAS nr:

942206-85-1

Purity:

98%

Molecular Weight:

655,61

SMILES:

CC(C)C[C@H](NC(=O)c1cc2ccccc2s1)C(=O)N1CCN(CC1)C(=O)[C@H](CO)NS(=O)(=O)c1ccc(Cl)cc1Cl

Formula:

C28H32Cl2N4O6S2

Pathway:

Membrane transporter/Ion channel,Metabolism,Membrane transporter/Ion channel

Target:

TRP/TRPV Channel,Calcium Channel,Calcium Channel