Bioactivity:

CTAP TFA is a potent, highly selective, and brain penetrant �antagonist of _-opioid receptor with IC50 of 3.5 nM.�It displays over 1200-fold selectivity over _ opioid (IC50=4500 nM) and somatostatin receptors.�CTAP TFA can be used for the study of L-DOPA-

CAS nr:

TP2050L

Purity:

98%

Molecular Weight:

SMILES:

CC(O)C1C(NC(C(NC(C(N)=O)C(O)C)=O)C(C)(C)SSCC(NC(C(N)CC2=CC=CC=C2)=O)C(NC(CC3=CC=C(O)C=C3)C(NC(CC4=CNC5=CC=CC=C54)C(NC(CCC/N=C(N)\N)C(N1)=O)=O)=O)=O)=O.O=C(O)C(F)(F)F

Formula:

Pathway:

Endocrinology/Hormones,Neuroscience,GPCR/G Protein

Target:

Opioid Receptor,Opioid Receptor,Opioid Receptor