Bioactivity:

CGP71683 is a competitive neuropeptide Y5 receptor antagonist (Ki: 1.3 nM) and shows no obvious activity at Y1 receptor (Ki >4000 nM) and Y2 receptor (Ki: 200 nM) in cell membranes.

CAS nr:

192322-50-2

Purity:

98%

Molecular Weight:

512,07

SMILES:

Cl.Nc1nc(NC[C@H]2CC[C@H](CNS(=O)(=O)c3cccc4ccccc34)CC2)nc2ccccc12

Formula:

C26H30ClN5O2S

Pathway:

GPCR/G Protein,Neuroscience

Target:

Neuropeptide Y Receptor,Neuropeptide Y Receptor