Bioactivity:

A-317491 is a non-nucleotide P2X3 ( Ki: 22 nM) and P2X2/3 receptor (Ki: 9 nM) antagonist, which inhibits calcium flux mediated by the receptors.

CAS nr:

475205-49-3

Purity:

98%

Molecular Weight:

565,57

SMILES:

O=C(C1=CC(C(N(CC2=CC=CC(OC3=CC=CC=C3)=C2)[C@H]4CCCC5=C4C=CC=C5)=O)=C(C(O)=O)C=C1C(O)=O)O

Formula:

C33H27NO8

Pathway:

Membrane transporter/Ion channel,Neuroscience

Target:

P2X Receptor,P2 Receptor