GSK-5959 T1972
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
GSK-5959 is an effective, specific and cell permeable BRPF1 bromodomain inhibitor (IC50: ~80 nM). The selectivity of GSK-5959 for BRPF1 is >100-fold over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains.
CAS nr:
901245-65-6
Purity:
98%
Molecular Weight:
394,47
SMILES:
COc1ccccc1C(=O)Nc1c(cc2n(C)c(=O)n(C)c2c1)N1CCCCC1
Formula:
C22H26N4O3
Pathway:
Chromatin/Epigenetic
Target:
Epigenetic Reader Domain
