Bioactivity:

CSRM617 is a selective small molecule inhibitor of the transcription factor ONECUT2 (OC2, the main regulator of androgen receptor). The Kd in SPR analysis is 7.43 uM, which can directly bind to the OC2-HOX domain. CSRM617 induces apoptosis by cleaving the

CAS nr:

787504-88-5

Purity:

98%

Molecular Weight:

255,23

SMILES:

N[C@@H](CO)C(N/N=C/C1=CC=C(O)C(O)=C1O)=O

Formula:

C10H13N3O5

Pathway:

Others

Target:

Others