Bioactivity:

JP1302 dihydrochloride is a selective, high affinity antagonist of the alpha2C-adrenoceptor (_2C-adrenoceptor), with a Ki (binding affinity) value of 28 nM and a Kb value (antagonist activity) of 16 nM.

CAS nr:

1259314-65-2

Purity:

98%

Molecular Weight:

441,4

SMILES:

CN1CCN(C2=CC=C(NC3=C(C=CC=C4)C4=NC5=CC=CC=C53)C=C2)CC1.[H]Cl.[H]Cl

Formula:

C24H26Cl2N4

Pathway:

Neuroscience,GPCR/G Protein

Target:

Adrenergic Receptor,Adrenergic Receptor