Bioactivity:

GKA50 stimulates insulin release from mouse islets of Langerhans and MIN6 cells. GKA50 shows significant glucose lowering in high fat fed female rats.�GKA50 is a potent glucokinase activator (EC50=33 nM at 5 mM glucose).

CAS nr:

851884-87-2

Purity:

98%

Molecular Weight:

464,51

SMILES:

O=C(C1=CC=C(NC(C2=CC(O[C@@H](C)CC3=CC=CC=C3)=CC(O[C@@H](C)COC)=C2)=O)N=C1)O

Formula:

C26H28N2O6

Pathway:

Others

Target:

Others