Bioactivity:

A922500 is an inhibitor for human and mouse DGAT-1 with IC50 of 7 nM and 24 nM, respectively, good selectivity over related acyltransferases, hERG, and a panel of anti-targets.

CAS nr:

959122-11-3

Purity:

98%

Molecular Weight:

428,48

SMILES:

OC(=O)[C@@H]1CCC[C@H]1C(=O)C1=CC=C(C=C1)C1=CC=C(NC(=O)NC2=CC=CC=C2)C=C1

Formula:

C26H24N2O4

Pathway:

Proteases/Proteasome,Metabolism,Metabolism

Target:

Acyltransferase,Transferase,Acyltransferase