Dbet57 T5440
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
dBET57 is heterobifunctional degrader of BRD4 based on the PROTAC technology, exhibits significant degradation of BRD4BD1 with a DC50/5h of 500 nM ,and�inactive on BRD4BD2
CAS nr:
1883863-52-2
Purity:
98%
Molecular Weight:
699,18
SMILES:
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCNc1cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c13)c1nnc(C)n-21)c1ccc(Cl)cc1
Formula:
C34H31ClN8O5S
Pathway:
Chromatin/Epigenetic
Target:
Epigenetic Reader Domain
