Bioactivity:

GLL398 is an oral selective estrogen receptor down-regulating agent that strongly binds to ER_ (IC50 =1.14 nM) and effectively degrades ER_ in MCF-7 breast cancer cells (IC50 = 0.21 _M).

CAS nr:

2077980-83-5

Purity:

98%

Molecular Weight:

398,27

SMILES:

O=C(O)/C=C/C1=CC=C(/C(C2=CC=C(B(O)O)C=C2)=C(C3=CC=CC=C3)\CC)C=C1

Formula:

C25H23BO4

Pathway:

Target: