Bioactivity:

AP5 is a potent and selective agonist for the GPR40 receptor with positive allosteric modulation of endogenous ligands (AgoPAM). AP5 demonstrates a rat hIP1 EC50 of 0.49 nM against the GPR40 receptor.

CAS nr:

1623194-37-5

Purity:

98%

Molecular Weight:

461,52

SMILES:

FC1=CC(C2=CC(OC)=NC=C2)=CC=C1[C@@H]3CCC(C=CC([C@H](C4CC4)[C@H](C)C(O)=O)=C5)=C5O3

Formula:

C28H28FNO4

Pathway:

Others

Target:

Others