Bioactivity:

ERK-IN-2 might lead to off-target toxicity and/or off-target activity at dose >10 _M.ERK-IN-2 is a potent, highly seletive and orally active ERK2 inhibitor probe with an IC50 value of 1.8 nM.

CAS nr:

T11225

Purity:

98%

Molecular Weight:

347,8

SMILES:

OCC1=NC(NC(N[C@H](C)C2=CC=CC=C2)=O)=CC3=C1C=NN3.[H]Cl

Formula:

C16H18ClN5O2

Pathway:

MAPK

Target:

ERK