Bioactivity:

Desmethyl cariprazine is a Cariprazine active metabolite. Cariprazine, an antipsychotic drug candidate, shows a high affinity for the D3 (Ki: 0.085 nM) and D2 (Ki: 0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (2.6 nM).

CAS nr:

839712-15-1

Purity:

98%

Molecular Weight:

413,38

SMILES:

O=C(NC)N[C@@H]1CC[C@@H](CCN2CCN(C3=CC=CC(Cl)=C3Cl)CC2)CC1

Formula:

C20H30Cl2N4O

Pathway:

GPCR/G Protein,Neuroscience,GPCR/G Protein,Neuroscience

Target:

5-HT Receptor,5-HT Receptor,Dopamine Receptor,Dopamine Receptor