Bioactivity:

CS-003 free base (CS-003) is a triple tachykinin receptor antagonist with high affinity for human (neurokinin) NK1, NK2 and NK3 receptors, with Ki values of 2.3 nM and 0.54 nM, respectively And 0.74 nM. CS-003 free base (CS-003) has therapeutic effects on

CAS nr:

191672-52-3

Purity:

98%

Molecular Weight:

673,65

SMILES:

O=C(N1C[C@@](CCN2CCC3(CC2)C4=CC=CC=C4C[S@@]3=O)(C5=CC=C(Cl)C(Cl)=C5)OCC1)C6=CC(OC)=C(OC)C(OC)=C6

Formula:

C34H38Cl2N2O6S

Pathway:

Neuroscience,GPCR/G Protein

Target:

Neurokinin receptor,Neurokinin receptor