Bioactivity:

BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM and it also is selective and potent for CYP3A4 activity with an EC50 of 13 _M.

CAS nr:

1197420-05-5

Purity:

98%

Molecular Weight:

468,95

SMILES:

ClC1=CC=C(C2=CC(N=CN(C3=CC(OC)=C(OC[C@H](O)C4CC4)C=C3)C5=O)=C5S2)C=C1

Formula:

C24H21ClN2O4S

Pathway:

Metabolism

Target:

P450