Bioactivity:

L-798106 is a highly selective prostanoid EP3 receptor antagonist (Ki=0.3 nM). It also has micromolar activities at EP4, EP1, and EP2 receptors (Ki: 916 nM, >5000 nM, and >5000 nM at EP4, EP1, and EP2, respectively).

CAS nr:

244101-02-8

Purity:

98%

Molecular Weight:

536,44

SMILES:

O=C(NS(=O)(C1=CC(Br)=CC=C1OC)=O)/C=C/C2=CC=CC=C2CC3=CC=C4C=CC=CC4=C3

Formula:

C27H22BrNO4S

Pathway:

GPCR/G Protein,Immunology/Inflammation

Target:

Prostaglandin Receptor,Prostaglandin Receptor