Bioactivity:

BET-IN-6 is an effective and high-affinity inhibitor of BRD2/BRD4. It is the ligand for target protein BRD2/4 and is used for the synthesis of PROTAC BRD2/BRD4 degrader-1.

CAS nr:

T10522

Purity:

98%

Molecular Weight:

440,47

SMILES:

O=C(O)CCC1=CC2=C(C=CC(N(C3=O)C)=C2C3=C1)NS(=O)(C4=CC=CC=C4OC)=O

Formula:

C22H20N2O6S

Pathway:

Chromatin/Epigenetic

Target:

Epigenetic Reader Domain