Bioactivity:

DYRKs-IN-2 has antitumor activity. DYRKs-IN-2 is a potent DYRKs inhibitor with IC50s of 30.6 nM and 12.8 nM for DYRK1B and DYRK1A, respectively.

CAS nr:

1386980-04-6

Purity:

98%

Molecular Weight:

632,16

SMILES:

O=C(C1=CC2=CN=C(NCCCN3CCN(C)CC3)N=C2NC1=O)NC4=CC(C(NC(C5=CC=CC=C5)CCN)=O)=CC=C4Cl

Formula:

C32H38ClN9O3

Pathway:

Tyrosine Kinase/Adaptors,Cell Cycle/Checkpoint

Target:

DYRK,DYRK