PF 429242 T4317
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
PF-429242 is a competitive inhibitor of sterol regulatory element-binding protein (SREBP) site 1 protease (IC50 = 0.175 _M). It is selective for site 1 protease against a panel of serine proteases. PF-429242 inhibits rate of cholesterol synthesis in CHO c
CAS nr:
947303-87-9
Purity:
98%
Molecular Weight:
482,49
SMILES:
Cl.Cl.CCN(CC)Cc1ccc(cc1)C(=O)N(CCc1ccccc1OC)[C@@H]1CCNC1
Formula:
C25H35N3O2�2HCl
Pathway:
Metabolism,Membrane transporter/Ion channel
Target:
Lipid,NPC1L1
