Bioactivity:

ASP6432 is an antagonist of type 1 lysophosphatidic acid receptor (LPA1). For human LPA1 and rat LPA1, the IC50s are 11 nM and 30 nM , respectively.

CAS nr:

1282549-08-9

Purity:

98%

Molecular Weight:

598,78

SMILES:

O=C(C1=CSC(CN(C(C2=CC(OC)=C(C)C(OC)=C2)=O)CCCC3=CC=CC=C3)=N1)[N-]S(=O)(NCC)=O.[K+]

Formula:

C26H31KN4O6S2

Pathway:

GPCR/G Protein

Target:

LPA Receptor